Andrés A. Trabanco : rechercher sur Z-Library

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1

Synthesis, Evaluation, and Radiolabeling of New Potent Positive Allosteric Modulators of the Metabotropic Glutamate Receptor 2 as Potential Tracers for Positron Emission Tomography Imaging

Andrés, José-Ignacio, Alcázar, Jesús, Cid, José María, De Angelis, Meri, Iturrino, Laura, Langlois, Xavier, Lavreysen, Hilde, Trabanco, Andrés A., Celen, Sofie, Bormans, Guy

Journal:

Journal of Medicinal Chemistry

Année:

2012

Langue:

english

Fichier:

PDF, 561 KB

english, 2012

2

Dihydrothiazolopyridone Derivatives as a Novel Family of Positive Allosteric Modulators of the Metabotropic Glutamate 5 (mGlu 5 ) Receptor

Bartolomé-Nebreda, José Manuel, Conde-Ceide, Susana, Delgado, Francisca, Iturrino, Laura, Pastor, Joaquín, Pena, Miguel Ángel, Trabanco, Andrés A., Tresadern, Gary, Wassvik, Carola M., Stauffer, Shaun

Journal:

Journal of Medicinal Chemistry

Année:

2013

Langue:

english

Fichier:

PDF, 1.35 MB

english, 2013

3

Diastereoselective Synthesis of 2-Phenyl-3-(trifluoromethyl)piperazines as Building Blocks for Drug Discovery

Sánchez-Roselló, María, Delgado, Oscar, Mateu, Natalia, Trabanco, Andrés A., Van Gool, Michiel, Fustero, Santos

Journal:

Journal of Organic Chemistry

Année:

2014

Langue:

english

Fichier:

PDF, 361 KB

english, 2014

4

Pharmacological Characterization of JNJ-40068782, a New Potent, Selective, and Systemically Active Positive Allosteric Modulator of the mGlu2 Receptor and Its Radioligand [3H]JNJ-40068782

Lavreysen, H., Langlois, X., Ahnaou, A., Drinkenburg, W., te Riele, P., Biesmans, I., Van der Linden, I., Peeters, L., Megens, A., Wintmolders, C., Cid, J. M., Trabanco, A. A., Andres, J. I., Dautzenb

Journal:

Journal of Pharmacology and Experimental Therapeutics

Année:

2013

Langue:

english

Fichier:

PDF, 1.62 MB

english, 2013

5

1,3,5-Trisubstituted Pyrazoles as Potent Negative Allosteric Modulators of the mGlu 2/3 Receptors

Van Gool, Michiel, Alonso De Diego, Sergio A., Delgado, Oscar, Trabanco, Andrés A., Jourdan, Fabrice, Macdonald, Gregor J., Somers, Marijke, Ver Donck, Luc

Journal:

Année:

2017

Langue:

english

Fichier:

PDF, 2.17 MB

english, 2017

6

Hydrochlorofluoromethylation of unactivated alkenes with chlorofluoroacetic acid

Meyer, Claudio F., Hell, Sandrine M., Sap, Jeroen B.I., Misale, Antonio, Peschiulli, Aldo, Oehlrich, Daniel, Trabanco, Andrés A., Gouverneur, Véronique

Journal:

Année:

2019

Langue:

english

Fichier:

PDF, 648 KB

english, 2019

7

2- and 3-Haloalkoxy Fischer Carbene Complexes of Chromium as Synthons for either Hydroxycyclopropanation or Oxaspirocyclopropanation of Alkenes

José Barluenga, Salomé López, Andrés A. Trabanco, Josefa Flórez

Journal:

Chemistry - A European Journal

Année:

2001

Langue:

english

Fichier:

PDF, 139 KB

english, 2001

8

Mononuclear Biscarbene Complexes by Direct Nucleophile Addition to a CO Ligand of Fischer Arylcarbene Complexes

José Barluenga, Andrés A. Trabanco, Iván Pérez-Sánchez, Raquel De la Campa, Josefa Flórez, Santiago García-Granda, Ángel Aguirre

Journal:

Chemistry - A European Journal

Année:

2008

Langue:

english

Fichier:

PDF, 212 KB

english, 2008

9

ChemInform Abstract: Asymmetric Benzopentaannulation from Tungsten ((-)-Menthyloxy)(aryl)carbene Complexes, Alkynyllithiums, and Methyl Triflate.

Jose Barluenga, Andres A. Trabanco, Josefa Florez, Santiago Garcia-Granda, Maria-Amparo LLorca

Journal:

Année:

1999

Langue:

english

Fichier:

PDF, 37 KB

english, 1999

10

ChemInform Abstract: A seco-Porphyrazine: Superb Sensitizer for Singlet Oxygen Generation and Endoperoxide Synthesis.

Andres A. Trabanco, Antonio Garrido Montalban, Garry Rumbles, Anthony G. M. Barrett, Brian M. Hoffman

Journal:

Année:

2000

Fichier:

PDF, 32 KB

2000

11

ChemInform Abstract: Diastereoselective Intermolecular Cyclopropanation of Simple Alkenes by Fischer Alkenyl and Heteroaryl Carbene Complexes of Chromium: Scope and Limitations.

Jose Barluenga, Salome Lopez, Andres A. Trabanco, Alvaro Fernandez-Acebes, Josefa Florez

Journal:

Année:

2000

Fichier:

PDF, 34 KB

2000

12

ChemInform Abstract: 2- and 3-Haloalkoxy Fischer Carbene Complexes of Chromium as Synthons for Either Hydroxycyclopropanation or Oxaspirocyclopropanation of Alkenes.

Jose Barluenga, Salome Lopez, Andres A. Trabanco, Josefa Florez

Journal:

Année:

2002

Fichier:

PDF, 32 KB

2002

13

Selective α-Monoallylation of Phenyl Ketones and Benzocycloalkanones under Microwave Irradiation.

Jose M. Cid, Juan L. Romera, Andres A. Trabanco

Journal:

Année:

2004

Fichier:

PDF, 104 KB

2004

14

Synthesis of 2-N,N-Dimethylaminomethyl-2,3,3a,12b-tetrahydrodibenzo[b,f]furo [2,3-d]oxepin Derivatives as Potential Anxiolytic Agents.

Andres Avelino Trabanco, Jose Manuel Alonso, Jose Ignacio Andres, Jose Maria Cid, Javier Fernandez, Laura Iturrino, Anton Megens

Journal:

Année:

2004

Langue:

english

Fichier:

PDF, 146 KB

english, 2004

15

Potassium Iodide Catalyzed Monoalkylation of Anilines under Microwave Irradiation.

Juan L. Romera, Jose M. Cid, Andres A. Trabanco

Journal:

Année:

2005

Fichier:

PDF, 28 KB

2005

16

Synthesis of 2-N,N-Dimethylaminomethyl-2,3,3a,12b-tetrahydrodibenzo[b,f]furo [2,3-d]oxepine Derivatives as Potential Anxiolytic Agents. Part 2. Substitutions by Methyl Groups on the Tetrahydrofuran Ring.

Andres A. Trabanco, Jose M. Alonso, Jose M. Cid, Luis Miguel Font, Anton Megens

Journal:

Année:

2005

Fichier:

PDF, 41 KB

2005

17

Novel 2-N,N-Dimethylaminomethyl-2,3,3a,12b-tetrahydrodibenzo[b,f]furo [2,3-d]oxepin Derivatives Displaying Combined Norepinephrine Reuptake Inhibition and 5-HT2A/2C Receptor Antagonism.

Jose M. Bartolome, Ana Alcudia, Jose I. Andres, Jose M. Cid, Mercedes Garcia, Anton Megens, Miguel A. Toledo, Andres A. Trabanco

Journal:

Année:

2005

Fichier:

PDF, 23 KB

2005

18

ChemInform Abstract: Microwave-Assisted N-Debenzylation of Amides with Triflic Acid.

Frederik Rombouts, Dennis Franken, Carolina Martinez-Lamenca, Mirielle Braeken, Chiara Zavattaro, Jinsheng Chen, Andres A. Trabanco

Journal:

Année:

2010

Fichier:

PDF, 31 KB

2010

19

Synthesis and structure–activity relationship of 2-(aminoalkyl)-3,3a,8,12b-tetrahydro-2H-dibenzocyclohepta[1,2-b]furan derivatives: a novel series of 5-HT2A/2C receptor antagonists

José Cid, José M. Alonso, José I. Andrés, Javier Fernández, Pilar Gil, Laura Iturrino, Encarna Matesanz, Theo F. Meert, Anton Megens, Victor K. Sipido, Andrés A. Trabanco

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2004

Langue:

english

Fichier:

PDF, 335 KB

english, 2004

20

Novel 2-N,N-dimethylaminomethyl-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepin derivatives displaying combined norepinephrine reuptake inhibition and 5-HT2A/2C receptor antagonism

José M. Bartolomé, Ana Alcudia, José I. Andrés, José M. Cid, Mercedes García, Anton Megens, Miguel A. Toledo, Andrés A. Trabanco

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2005

Langue:

english

Fichier:

PDF, 206 KB

english, 2005

21

4-Phenyl-4-[1H-imidazol-2-yl]-piperidine derivatives, a novel class of selective δ-opioid agonists

Andrés A. Trabanco, Shirley Pullan, José M. Alonso, Rosa M. Alvarez, José I. Andrés, Inge Boeckx, Javier Fernández, Antonio Gómez, Laura Iturrino, Frans E. Janssens, Joseph E. Leenaerts, Ana I. De Luc

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2006

Langue:

english

Fichier:

PDF, 117 KB

english, 2006

22

4-Phenyl-4-[1H-imidazol-2-yl]-piperidine derivatives as non-peptidic selective δ-opioid agonists with potential anxiolytic/antidepressant properties. Part 2

Andrés A. Trabanco, Nancy Aerts, Rosa M. Alvarez, José I. Andrés, Inge Boeckx, Javier Fernández, Antonio Gómez, Frans E. Janssens, Joseph E. Leenaerts, Ana I. De Lucas, Encarna Matesanz, Thomas Steckl

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2007

Langue:

english

Fichier:

PDF, 170 KB

english, 2007

23

New positive allosteric modulators of the metabotropic glutamate receptor 2 (mGluR2): Identification and synthesis of N-propyl-8-chloro-6-substituted isoquinolones

Andrés A. Trabanco, Guillaume Duvey, José María Cid, Gregor J. Macdonald, Philippe Cluzeau, Vanthea Nhem, Rocco Furnari, Nadia Behaj, Géraldine Poulain, Terry Finn, Hilde Lavreysen, Sonia Poli, Alexan

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2011

Langue:

english

Fichier:

PDF, 1.77 MB

english, 2011

24

Selective α-monoallylation of phenyl ketones and benzocycloalkanones under microwave irradiation

José M. Cid, Juan L. Romera, Andrés A. Trabanco

Journal:

Tetrahedron Letters

Année:

2004

Langue:

english

Fichier:

PDF, 287 KB

english, 2004

25

Potassium iodide catalysed monoalkylation of anilines under microwave irradiation

Juan L. Romera, José M. Cid, Andrés A. Trabanco

Journal:

Tetrahedron Letters

Année:

2004

Langue:

english

Fichier:

PDF, 289 KB

english, 2004

26

Microwave-assisted N-debenzylation of amides with triflic acid

Frederik Rombouts, Dennis Franken, Carolina Martínez-Lamenca, Mirielle Braeken, Chiara Zavattaro, Jinsheng Chen, Andrés A. Trabanco

Journal:

Tetrahedron Letters

Année:

2010

Langue:

english

Fichier:

PDF, 416 KB

english, 2010

27

Synthesis of 2-N,N-dimethylaminomethyl-2,3,3a,12b-tetrahydrodibenzo[b,f]furo[2,3-d]oxepine derivatives as potential anxiolytic agents. Part 2: substitutions by methyl groups on the tetrahydrofuran ring

Andrés A. Trabanco, José M. Alonso, José M. Cid, Luis Miguel Font, Anton Megens

Journal:

Année:

2005

Langue:

english

Fichier:

PDF, 333 KB

english, 2005

28

Design and Synthesis of a Novel Series of Bicyclic Heterocycles As Potent γ-Secretase Modulators

Bischoff, Francois, Berthelot, Didier, De Cleyn, Michel, Macdonald, Gregor, Minne, Garrett, Oehlrich, Daniel, Pieters, Serge, Surkyn, Michel, Trabanco, Andrés A., Tresadern, Gary, Van Brandt, Sven, Ve

Journal:

Journal of Medicinal Chemistry

Année:

2012

Langue:

english

Fichier:

PDF, 2.17 MB

english, 2012

29

Synthesis and Reactions of Aminoporphyrazines with Annulated Five- and Seven-Membered Rings

Suhling, Klaus, Phillips, David, White, Andrew J. P., Williams, David J., Baum, Sven M., Trabanco, Andrés A., Montalban, Antonio Garrido, Micallef, Aaron S., Zhong, Chang, Meunier, Hubert G.

Journal:

Journal of Organic Chemistry

Année:

2003

Langue:

english

Fichier:

PDF, 271 KB

english, 2003

30

A practical entry to β-aryl-β-alkyl amino alcohols: application to the synthesis of a potent BACE1 inhibitor

Delgado, Oscar, Monteagudo, Antonio, Van Gool, Michiel, Trabanco, Andrés A., Fustero, Santos

Journal:

Organic & Biomolecular Chemistry

Année:

2012

Langue:

english

Fichier:

PDF, 219 KB

english, 2012

31

Regioselective Preparation of 3-Alkoxy-4,5-difluoroanilines by S N Ar

Van Brandt, Sven, Rombouts, Frederik J. R., Martínez-Lamenca, Carolina, Leenaerts, Jos, Rauws, Tom R. M., Trabanco, Andrés A.

Journal:

European Journal of Organic Chemistry

Année:

2012

Langue:

english

Fichier:

PDF, 541 KB

english, 2012

32

Fluorous-Tagged Carbamates for the Pd-Catalyzed Amination of Aryl Halides

Trabanco, Andrés A., Vega, Juan A., Fernández, M. Alejandro

Journal:

Journal of Organic Chemistry

Année:

2007

Langue:

english

Fichier:

PDF, 155 KB

english, 2007

33

mGluR2 positive allosteric modulators: a patent review (2009 – present)

Trabanco, Andrés A, Cid, José María

Journal:

Expert Opinion on Therapeutic Patents

Année:

2013

Langue:

english

Fichier:

PDF, 1.71 MB

english, 2013

34

Design and synthesis of bicyclic heterocycles as potent γ-secretase modulators

Oehlrich, Daniel, Rombouts, Frederik J.R., Berthelot, Didier, Bischoff, François P., De Cleyn, Michel A.J., Jaroskova, Libuse, Macdonald, Gregor, Mercken, Marc, Surkyn, Michel, Trabanco, Andrés A., Tr

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2013

Langue:

english

Fichier:

PDF, 1.47 MB

english, 2013

35

Asymmetric Conjugate Nucleophilic Addition of Organolithiums to Chromium (Menthyloxy)(aryl)carbene Complexes

Barluenga, José, Trabanco, Andrés A., Flórez, Josefa, García-Granda, Santiago, Martín, Eduardo

Journal:

Journal of the American Chemical Society

Année:

1996

Langue:

english

Fichier:

PDF, 203 KB

english, 1996

36

A General Synthesis of α-Trifluoromethylstyrenes through Palladium-Catalyzed Cross-Couplings with 1,1,1-Trifluoroacetone Tosylhydrazone

Jiménez-Aquino, Agustín, Vega, Juan A., Trabanco, Andrés A., Valdés, Carlos

Journal:

Advanced Synthesis & Catalysis

Année:

2014

Langue:

english

Fichier:

PDF, 267 KB

english, 2014

37

Discovery of a new series of [1,2,4]triazolo[4,3-a]quinoxalines as dual phosphodiesterase 2/phosphodiesterase 10 (PDE2/PDE10) inhibitors

Andrés, José-Ignacio, Buijnsters, Peter, De Angelis, Meri, Langlois, Xavier, Rombouts, Frederik, Trabanco, Andrés A., Vanhoof, Greet

Journal:

Bioorganic & Medicinal Chemistry Letters

Année:

2013

Langue:

english

Fichier:

PDF, 5.60 MB

english, 2013

38

QSAR design of triazolopyridine mGlu2 receptor positive allosteric modulators

Tresadern, Gary, Cid, José-Maria, Trabanco, Andrés A.

Journal:

Journal of Molecular Graphics and Modelling

Année:

2014

Langue:

english

Fichier:

PDF, 2.01 MB

english, 2014

39

Discovery of New Tetracyclic Tetrahydrofuran Derivatives as Potential Broad-Spectrum Psychotropic Agents

Fernández, Javier, Alonso, José M., Andrés, José I., Cid, José M., Díaz, Adolfo, Iturrino, Laura, Gil, Pilar, Megens, Anton, Sipido, Victor K., Trabanco, Andrés A.

Journal:

Journal of Medicinal Chemistry

Année:

2005

Langue:

english

Fichier:

PDF, 85 KB

english, 2005

40

Diastereoselective Cyclopropanation of Simple Alkenes by 2-Phenyl- and 2-Ferrocenylalkenyl Fischer Carbene Complexes of Chromium

Barluenga, José, Fernández-Acebes, Alvaro, Trabanco, Andrés A., Flórez, Josefa

Journal:

Journal of the American Chemical Society

Année:

1997

Langue:

english

Fichier:

PDF, 142 KB

english, 1997

41

Imidazo[1,2- a ]pyridines: Orally Active Positive Allosteric Modulators of the Metabotropic Glutamate 2 Receptor

Trabanco, Andrés A., Tresadern, Gary, Macdonald, Gregor J., Vega, Juan Antonio, de Lucas, Ana Isabel, Matesanz, Encarnación, García, Aránzazu, Linares, María Lourdes, Alonso de Diego, Sergio A., Alons

Journal:

Journal of Medicinal Chemistry

Année:

2012

Langue:

english

Fichier:

PDF, 1.55 MB

english, 2012

42

Asymmetric Benzopentaannulation from Tungsten ((−)-Menthyloxy)(aryl)carbene Complexes, Alkynyllithiums, and Methyl Triflate

Barluenga, José, Trabanco, Andrés A., Flórez, Josefa, García-Granda, Santiago, LLorca, María-Amparo

Journal:

Journal of the American Chemical Society

Année:

1998

Langue:

english

Fichier:

PDF, 127 KB

english, 1998

43

Diastereoselective Intermolecular Cyclopropanation of Simple Alkenes by Fischer Alkenyl and Heteroaryl Carbene Complexes of Chromium: Scope and Limitations

Barluenga, José, López, Salomé, Trabanco, Andrés A., Fernández-Acebes, Alvaro, Flórez, Josefa

Journal:

Journal of the American Chemical Society

Année:

2000

Langue:

english

Fichier:

PDF, 190 KB

english, 2000

44

Structure-Based Design of a Potent, Selective, and Brain Penetrating PDE2 Inhibitor with Demonstrated Target Engagement

Buijnsters, Peter, De Angelis, Meri, Langlois, Xavier, Rombouts, Frederik J. R., Sanderson, Wendy, Tresadern, Gary, Ritchie, Alison, Trabanco, Andrés A., VanHoof, Greet, Roosbroeck, Yves Van, Andrés,

Journal:

ACS Medicinal Chemistry Letters

Année:

2014

Langue:

english

Fichier:

PDF, 372 KB

english, 2014

45

Pyrido[4,3- e ][1,2,4]triazolo[4,3- a ]pyrazines as Selective, Brain Penetrant Phosphodiesterase 2 (PDE2) Inhibitors

Rombouts, Frederik J. R., Tresadern, Gary, Buijnsters, Peter, Langlois, Xavier, Tovar, Fulgencio, Steinbrecher, Thomas B., Vanhoof, Greet, Somers, Marijke, Andrés, José-Ignacio, Trabanco, Andrés A.

Journal:

ACS Medicinal Chemistry Letters

Année:

2015

Langue:

english

Fichier:

PDF, 1.29 MB

english, 2015

46

Pharmacological and pharmacokinetic properties of JNJ-40411813, a positive allosteric modulator of the mGlu2 receptor

Lavreysen, Hilde, Ahnaou, Abdellah, Drinkenburg, Wilhelmus, Langlois, Xavier, Mackie, Claire, Pype, Stefan, Lütjens, Robert, Le Poul, Emmanuel, Trabanco, Andrés A., Nuñez, José María Cid

Journal:

Pharmacology Research & Perspectives

Année:

2015

Langue:

english

Fichier:

PDF, 840 KB

english, 2015

47

N-bridged 5,6-bicyclic pyridines: Recent applications in central nervous system disorders

Delgado, Oscar, Delgado, Francisca, Vega, Juan Antonio, Trabanco, Andrés A.

Journal:

European Journal of Medicinal Chemistry

Année:

2015

Langue:

english

Fichier:

PDF, 1.80 MB

english, 2015

48

Benzazaborinines as Novel Bioisosteric Replacements of Naphthalene: Propranolol as an Example

Rombouts, Frederik J. R., Tovar, Fulgencio, Austin, Nigel, Tresadern, Gary, Trabanco, Andrés A.

Journal:

Journal of Medicinal Chemistry

Année:

2015

Langue:

english

Fichier:

PDF, 1.21 MB

english, 2015

49

Cover Picture: A Versatile Approach to CF 3 -Containing 2-Pyrrolidones by Tandem Michael Addition-Cyclization: Exemplification in the Synthesis of Amidine Class BACE1 Inhibitors (Chem. Eur. J. 33/2015)

Mateu, Natalia, Ciordia, Myriam, Delgado, Oscar, Sánchez-Roselló, María, Trabanco, Andrés A., Van Gool, Michiel, Tresadern, Gary, Pérez-Benito, Laura, Fustero, Santos

Journal:

Chemistry - A European Journal

Année:

2015

Fichier:

PDF, 439 KB

2015

50

A Versatile Approach to CF 3 -Containing 2-Pyrrolidones by Tandem Michael Addition-Cyclization: Exemplification in the Synthesis of Amidine Class BACE1 Inhibitors

Mateu, Natalia, Ciordia, Myriam, Delgado, Oscar, Sánchez-Roselló, María, Trabanco, Andrés A., Van Gool, Michiel, Tresadern, Gary, Pérez-Benito, Laura, Fustero, Santos

Journal:

Chemistry - A European Journal

Année:

2015

Langue:

english

Fichier:

PDF, 1.16 MB

english, 2015